Discovery of Macrocyclic Myeloid Cell Leukemia 1 (Mcl-1) Inhibitors that Demonstrate Potent Cellular Efficacy and In Vivo Activity in a Mouse Solid Tumor Xenograft Model
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DOI: 10.1021/acs.jmedchem.5c01376
文献链接: https://pubs.acs.org/doi/10.1021/acs.jmedchem.5c01376
其他信息:
出版社: American Chemical Society (ACS)
作者: James C. Tarr; Kyuok Jeon; Nagarathanam Veerasamy; Martin Aichinger; James M. Salovich; Bin Zhao; John L. Sensintaffar; Heribert Arnhof; Tobias Wunberg; Danielle Sgubin; Allison Arnold; Rakesh H. Vekariya; Plamen P. Christov; Kwangho Kim; Julian Emanuel Fuchs; Pol Karier; Bodo Betzemeier; Mayme Van Meveren; Nagaraju Miriyala; Edward T. Olejniczak; Harald Engelhardt; Taekyu Lee; Darryl McConnell; Stephen W. Fesik
全文下载地址: https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5c01376