Discovery of LYA914, An Orally Bioavailable PROTAC Degrader Targeting the DNA Binding Domain of the Androgen Receptor for the Treatment of CRPC
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DOI: https://doi.org/10.1021/acs.jmedchem.5c01463
文献链接: https://pubs.acs.org/doi/10.1021/acs.jmedchem.5c01463
其他信息:
出版社: American Chemical Society (ACS)
作者: Yan Lv; Gaoxin Dai; Bowen Zhang; Chang Liu; Yiming Chen; Ling Ge; Sai Zhang; Siqi Zhang; Mengjun Ma; Shumin Ma; Chong Qin
全文下载地址: https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5c01463