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Discovery of a highly potent, selective, orally bioavailable inhibitor of KAT6A/B histone acetyltransferases with efficacy against KAT6A-high ER+ breast cancer复制

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DOI: DOI: 10.1016/j.chembiol.2023.07.005复制

文献链接: https://linkinghub.elsevier.com/retrieve/pii/S2451945623002349复制

其他信息:

出版社: Elsevier BV
作者: Shikhar Sharma; Chi-Yeh Chung; Sean Uryu; Jelena Petrovic; Joan Cao; Amanda Rickard; Nataliya Nady; Samantha Greasley; Eric Johnson; Oleg Brodsky; Showkhin Khan; Hui Wang; Zhenxiong Wang; Yong Zhang; Konstantinos Tsaparikos; Lei Chen; Anthony Mazurek; John Lapek; Pei-Pei Kung; Scott Sutton; Paul F. Richardson; Eric C. Greenwald; Shinji Yamazaki; Rhys Jones; Karen A. Maegley; Patrick Bingham; Hieu Lam; Alexandra E. Stupple; Aileen Kamal; Anderly Chueh; Anthony Cuzzupe; Benjamin J. Morrow; Bin Ren; Catalina Carrasco-Pozo; Chin Wee Tan; Dharmesh D. Bhuva; Elizabeth Allan; Elliot Surgenor; François Vaillant; Havva Pehlivanoglu; Hendrik Falk; James R. Whittle; Janet Newman; Joseph Cursons; Judy P. Doherty; Karen L. White; Laura MacPherson; Mark Devlin; Matthew L. Dennis; Meghan K. Hattarki; Melanie De Silva; Michelle A. Camerino; Miriam S. Butler; Olan Dolezal; Patricia Pilling; Richard Foitzik; Paul A. Stupple; H. Rachel Lagiakos; Scott R. Walker; Soroor Hediyeh-Zadeh; Stewart Nuttall; Sukhdeep K. Spall; Susan A. Charman; Theresa Connor; Thomas S. Peat; Vicky M. Avery; Ylva E. Bozikis; Yuqing Yang; Ming Zhang; Brendon J. Monahan; Anne K. Voss; Tim Thomas; Ian P. Street; Sarah-Jane Dawson; Mark A. Dawson; Geoffrey J. Lindeman; Melissa J. Davis; Jane E. Visvader; Thomas A. Paul

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