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Discovery of Potent and Brain-Penetrant Inverse Agonists for GPR61, an Orphan G Protein-Coupled Receptor复制

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DOI: https://doi.org/10.1021/acs.jmedchem.6c00081 复制

文献链接: https://pubs.acs.org/doi/10.1021/acs.jmedchem.6c00081复制

其他信息:

出版社: American Chemical Society (ACS)
作者: Ethan L. Fisher; Anne-Marie Dechert Schmitt; Jamison B. Tuttle; Ray Unwalla; Gabrielle H. Lovett; Bethany L. Kormos; Karen J. Coffman; Dahui Zhou; Michael Moran; Jade Williams; Jun Xiao; Erik A. LaChapelle; Jean-Philippe Fortin; Abdul Q. Sheikh; Kimberly A. Stevens; Jimmy X. Kong; Emily A. G. Hughes; Ryan M. Esquejo; Stephanie Joaquim; Nalissa L. Amar; Danielle Archambault; Jeonifer Garren; Danna Breen; Srinath Jagarlapudi; Robert Dullea; Rebecca E. O’Connor; Erika Koslov-Davino; Ernesto Callegari; João M. Dias; Joshua A. Lees; Kris Borzilleri; Seungil Han; Jonathan Brooks; Felix F. Vajdos; Ashish Goyal; Lei Zhang; Yuan Zhang
全文下载地址: https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.6c00081

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