Structure activity relationship exploration of imidazo[1,2-a]pyridine series to reverse isoform selectivity and identify potent SIK1 selective inhibitors
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DOI: https://doi.org/10.1016/j.bmcl.2025.130397
文献链接: https://linkinghub.elsevier.com/retrieve/pii/S0960894X25003063
其他信息:
出版社: Elsevier BV
作者: Christophe Peixoto; Elsa De Lemos; Laëtitia Cherel; Gregory Newsome; Aurelie Dos Santos; Irena Ćaleta; Thomas Coudrat; Kenneth Goossens; Mia Jans; Reginald Brys; Steve De Vos; David Amantini; Juan-Miguel Jimenez; Nicolas Desroy