Discovery of Bis-Acyl Hydrazides as Potent and Bioavailable MTA-Cooperative PRMT5 Inhibitors: A Case Study of Leveraging the Deuterium Kinetic Isotope Effect
DOI: 10.1021/acs.jmedchem.5c02392
文献链接: https://pubs.acs.org/doi/10.1021/acs.jmedchem.5c02392
其他信息:
出版社: American Chemical Society (ACS)
作者: Laurent Debien; Megan K. Armstrong; Joshua D. Farr; Ryan D. Ferrao; Pancham Lal Gupta; Congrong Niu; Andrew J. Anderson; Phillip Benner; Ashleigh N. Bristol; Elbert Chin; Chienhung Chou; Yifan Deng; Xiaoyong Fu; Mina Gheiratmand; Sarah M. Hull; Joey Chao-I Hung; Ben June; Jung Hwa Kirschman; Hoa Le; Bhavna Malik; Michael L. Mitchell; Prasenjit Kumar Mukherjee; Shaina V. Nguyen; Gregory T. Notte; Jessica Orf; Daniel E. Roa; Rex Santos; Adam J. Schrier; Katie A. Spence; Radhakrishna Sura; Zheng-Yu Yang; Doris Zane; Ariel N. Zahabian; Tatiana Zavorotinskaya

