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Discovery of Branebrutinib (BMS-986195): A Strategy for Identifying a Highly Potent and Selective Covalent Inhibitor Providing Rapid in Vivo Inactivation of Bruton’s Tyrosine Kinase (BTK)复制

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DOI: 10.1021/acs.jmedchem.9b00167复制

文献链接: https://pubs.acs.org/doi/10.1021/acs.jmedchem.9b00167复制

其他信息:

出版社: American Chemical Society (ACS)
作者: Scott H. Watterson; Qingjie Liu; Myra Beaudoin Bertrand; Douglas G. Batt; Ling Li; Mark A. Pattoli; Stacey Skala; Lihong Cheng; Mary T. Obermeier; Robin Moore; Zheng Yang; Rodney Vickery; Paul A. Elzinga; Lorell Discenza; Celia D’Arienzo; Kathleen M. Gillooly; Tracy L. Taylor; Claudine Pulicicchio; Yifan Zhang; Elizabeth Heimrich; Kim W. McIntyre; Qian Ruan; Richard A. Westhouse; Ian M. Catlett; Naiyu Zheng; Charu Chaudhry; Jun Dai; Michael A. Galella; Andrew J. Tebben; Matt Pokross; Jianqing Li; Rulin Zhao; Daniel Smith; Richard Rampulla; Alban Allentoff; Michael A. Wallace; Arvind Mathur; Luisa Salter-Cid; John E. Macor; Percy H. Carter; Aberra Fura; James R. Burke; Joseph A. Tino

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