Discovery of CFT8634, a Potent, Selective, and Orally Bioavailable Heterobifunctional Degrader of BRD9
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DOI: https://doi.org/10.1021/acs.jmedchem.5c01317
文献链接: https://pubs.acs.org/doi/10.1021/acs.jmedchem.5c01317
其他信息:
出版社: American Chemical Society (ACS)
作者: Katrina L. Jackson; Ning Yin; Roman V. Agafonov; Prasoon Chaturvedi; Kyle Cole; Scott J. Eron; Andrew C. Good; June A. Hart; Minsheng He; Christina S. Henderson; Hongwei Huang; R. Jason Kirby; Linda Lee; Moses Moustakim; Christopher G. Nasveschuk; Andrew J. Phillips; Roy M. Pollock; Laura L. Poling; Gesine K. Veits; Jeremy Yap; Rhamy Zeid; Amro Ali; Adam S. Crystal; Eunju Hurh; Huan Liu; Riadh Lobbardi; Leonard Reyno; Stewart L. Fisher
全文下载地址: https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5c01317

