Optimization of 2,3-dihydrophthalazine-1,4-dione PARP inhibitor scaffold for nanomolar potency and specificity towards human PARP10
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DOI: https://doi.org/10.1016/j.ejmech.2025.118111
文献链接: https://linkinghub.elsevier.com/retrieve/pii/S0223523425008761
其他信息:
出版社: Elsevier BV
作者: Juho Alaviuhkola; Maria Giulia Nizi; Chiara Vagaggini; Chiara Sarnari; Barbara Lippok; Mirko M. Maksimainen; Chiara Bosetti; Saurabh S. Dhakar; Giuseppe Manfroni; Serena Massari; Elena Dreassi; Patricia Korn; Oriana Tabarrini; Lari Lehtiö