Discovery of 2-(Pyrazol-4-yl)-quinazolin-4(3H)-one Derivatives as Subnanomolar BRD4 BD2 Inhibitors with High Selectivity via a Bioisosterism Approach
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DOI: https://doi.org/10.1021/acs.jmedchem.5c00924
文献链接: https://pubs.acs.org/doi/10.1021/acs.jmedchem.5c00924
其他信息:
出版社: American Chemical Society (ACS)
作者: Shuxia Chen; Jichen Yang; Qiong Wu; Jiaqi Zhou; Hui Shen; Xiangyu Wang; Yong Xu; Pingyuan Wang; Chang-Yun Wang; Yansheng Ye; Zhiqing Liu
全文下载地址: https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5c00924