Discovery of AZD8421: A Potent CDK2 Inhibitor with Selectivity Against Other CDK Family Members and the Human Kinome
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DOI: https://doi.org/10.1021/acs.jmedchem.5c01478
文献链接: https://pubs.acs.org/doi/10.1021/acs.jmedchem.5c01478
其他信息:
出版社: American Chemical Society (ACS)
作者: Avipsa Ghosh; Afshan Ahmed; Konstantina Amoiradaki; Amber Y. S. Balazs; Bernard Barlaam; Michael Steven Bodnarchuk; Gavin W. Collie; Ian L. Dale; Christopher R. Denz; Lisa Drew; Scott D. Edmondson; Jun Fan; Stephen Fawell; Frederick W. Goldberg; Ariamala Gopalsamy; Michael Grondine; Grace Guo; Sudhir M. Hande; Holia Hatoum-Mokdad; Alexander W. Hird; Rachel Howells; Jessie Hao-Ru Hsu; Jessica Hudson; Anne Jackson; Michelle L. Lamb; Gillian M. Lamont; Scott Lamont; Phillip A. Lichtor; Lisa McWilliams; David Milne; Scott N. Mlynarski; Priyanka Narasimhan; Matthew F. Peters; Alexander Pflug; Hannah Kate Pollard; Meile Qin; Corinne Reimer; Kevin J. Robbins; James Robinson; Li Sha; Hongyao She; James E. Sheppeck; Baljinder Singh; Kun Song; Qibin Su; Reem Telmesani; Scott Throner; Christina Vasalou; Lei Wang; Yanjun Wang; David M. Wilson; Poppy Winlow; Wenzhan Yang; Tieguang Yao; Yun Zhang; Zirong Zhang; Diana Zindel; Jeffrey W. Johannes
全文下载地址: https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5c01478