Damage Incorporated: Discovery of the Potent, Highly Selective, Orally Available ATR Inhibitor BAY 1895344 with Favorable Pharmacokinetic Properties and Promising Efficacy in Monotherapy and in Combination Treatments in Preclinical Tumor Models
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DOI: https://doi.org/10.1021/acs.jmedchem.0c00369
文献链接: https://pubs.acs.org/doi/10.1021/acs.jmedchem.0c00369
其他信息:
出版社: American Chemical Society (ACS)
作者: Ulrich Lücking; Lars Wortmann; Antje M. Wengner; Julien Lefranc; Philip Lienau; Hans Briem; Gerhard Siemeister; Ulf Bömer; Karsten Denner; Martina Schäfer; Marcus Koppitz; Knut Eis; Florian Bartels; Benjamin Bader; Wilhelm Bone; Dieter Moosmayer; Simon J. Holton; Uwe Eberspächer; Joanna Grudzinska-Goebel; Christoph Schatz; Gesa Deeg; Dominik Mumberg; Franz von Nussbaum